Dual specificity receptor for uracil nucleotides and cysteinyl leukotrienes (CysLTs). Signals through G(i) and inhibition of adenylyl cyclase. May mediate brain damage by nucleotides and CysLTs following ischemia.
Paruchuri, Jiang, Feng, Francis, Plutzky, Boyce: "Leukotriene E4 activates peroxisome proliferator-activated receptor gamma and induces prostaglandin D2 generation by human mast cells." in: The Journal of biological chemistry, Vol. 283, Issue 24, pp. 16477-87, (2008) (PubMed).
Parravicini, Ranghino, Abbracchio, Fantucci: "GPR17: molecular modeling and dynamics studies of the 3-D structure and purinergic ligand binding features in comparison with P2Y receptors." in: BMC bioinformatics, Vol. 9, pp. 263, (2008) (PubMed).
Ciana, Fumagalli, Trincavelli, Verderio, Rosa, Lecca, Ferrario, Parravicini, Capra, Gelosa, Guerrini, Belcredito, Cimino, Sironi, Tremoli, Rovati, Martini, Abbracchio: "The orphan receptor GPR17 identified as a new dual uracil nucleotides/cysteinyl-leukotrienes receptor." in: The EMBO journal, Vol. 25, Issue 19, pp. 4615-27, (2006) (PubMed).
Aliases for GPR17 抗体
G protein-coupled receptor 17 (GPR17) 抗体 G protein-coupled receptor 17 (Gpr17) 抗体 AI853548 抗体 GPR17 抗体